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3D MOLECULAR STRUCTURAL DATABASE OF BIOACTIVE COMPOUNDS FROM
NATURAL PRODUCTS
IN THAILAND
ADVANCE SEARCH
Plant Search
Plant Thai name
Plant common name
Plant scientific name
Family
Location
AND
OR
Chemical Search
Structure name
CAS No.
Formula
Class
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OR
Biological activity Search
Physicochemical properties
Molecular weight(g/mol)
Num. Heavy atom
Num. Aromatic atom
Num. Rotatable bond
Num. H-bond acceptor
Num. H-bond donor
TPSA(Angstrom)
Log P
Water Solubility Class
Insoluble
Poorly soluble
Moderately soluble
Soluble
Very soluble
Highly soluble
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AND
OR
Pharmacokinetics
GI absorption
----
High
Low
BBB permeant
----
Yes
No
Pgp substrate
----
Yes
No
CYP inhibitor
----
Yes
No
Log Kp (skin permeation) (cm/s)
AND
OR
Druglikeness
Lipinski Num. violations
Ghose Num. violations
Veber Num. violations
Egan Num. violations
Muegge Num. violations
Bioavailability Score
AND
OR
Medicinal Chemistry
PAINS Num. of alerts
Brenk Num. of alerts
Leadlikeness Num. of violations
Synthetic Accessibility
AND
OR